Deposited model

PDB 4ARK|dpdb_0duxnz5d

Deposited model

CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN MAP KINASE KINASE 1 (MEK1) IN COMPLEX WITH A SMALL MOLECULE INHIBITOR AND ADP

Program
REFMAC 5.4.0062
Model type
Deposited
Purpose
Reference
Authors
Hartung, I.V., Hitchcock, M., Puehler, F., Neuhaus, R., Scholz, A., Hammer, S., Petersen, K., Siemeister, G., Brittain, D., Hillig, R.C.
Atoms
2,381
Residues
291
Protein chains
1
Unmodeled fraction
14.66%
Ligands
ADP, MG

Evaluations

R-work
0.172
R-free
0.211
Clashscore
9.2

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
DUAL SPECIFICITY MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1341
  • ConstructCATALYTIC DOMAIN, RESIDUES 62-393

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations