Rerefined model

PDB 6TPD|dpdb_1tagfxcg

Rerefined model

Fragment-based discovery of pyrazolopyridones as JAK1 inhibitors with excellent subtype selectivity

Program
PHENIX 2.0_5824
Model type
Multiconformer
Purpose
Refinement
Atoms
2,691
Residues
289
Protein chains
1
Alternate-location fraction
0%
Ligand
QZ8

Evaluations

R-work
0.249
R-free
0.302
Clashscore
12.3

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Tyrosine-protein kinase JAK2289
  • MutationsY1007F/Y1008F

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations