Deposited model

PDB 1EAS|dpdb_3db6qfgk

Deposited model

NONPEPTIDIC INHIBITORS OF HUMAN LEUKOCYTE ELASTASE. 3. DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY RELATIONSHIPS FOR A SERIES OF ORALLY ACTIVE 3-AMINO-6-PHENYLPYRIDIN-2-ONE TRIFLUOROMETHYL KETONES

Program
X-PLOR
Model type
Deposited
Purpose
Reference
Authors
Ceccarelli, C.
Atoms
1,995
Residues
240
Protein chains
1
Unmodeled fraction
0%
Ligands
NA, TFK

Evaluations

R-work
0.183
R-free
—
Clashscore
4.9

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
PORCINE PANCREATIC ELASTASE240—

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations