Deposited model

PDB 4UYH|dpdb_3hfl5lfs

Deposited model

N-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 1-((2R,4S)-2-methyl-4-(phenylamino)-6-(4-(piperidin-1-ylmethyl)phenyl)-3,4-dihydroquinolin-1(2H)-yl)ethanone

Program
REFMAC 5.6.0117
Model type
Deposited
Purpose
Reference
Authors
Chung, C., Bamborough, P., Gosmini, R.
Atoms
3,269
Residues
321
Protein chains
3
Unmodeled fraction
30.52%

Evaluations

R-work
0.171
R-free
0.203
Clashscore
5.9

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
BROMODOMAIN-CONTAINING PROTEIN 2154
  • ConstructN-TERMINAL BROMODOMAIN, RESIDUES 67-200

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations