Deposited model

PDB 5VZS|dpdb_avjm5967

Deposited model

BRD4-BD1 in complex with Cpd19 (3-(7-(difluoromethyl)-6-(1-methyl-1H-pyrazol-4-yl)-3,4-dihydroquinolin-1(2H)-yl)-N-methyl-1-(tetrahydro-2H-pyran-4-yl)-1,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridine-5-carboxamide)

Program
PHENIX dev_2747
Model type
Deposited
Purpose
Reference
Authors
Murray, J.M.
Atoms
2,358
Residues
254
Protein chains
2
Unmodeled fraction
19.11%

Evaluations

R-work
0.192
R-free
0.226
Clashscore
1.8

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Bromodomain-containing protein 4157
  • ConstructBRD4 Bromodomain-1, UNP residues 42-168

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations