Deposited model

PDB 1C5Z|dpdb_caol83ki

Deposited model

STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR

Program
X-PLOR 3.1
Model type
Deposited
Purpose
Reference
Authors
Katz, B.A., Mackman, R., Luong, C., Radika, K., Martelli, A., Sprengeler, P.A., Wang, J., Chan, H., Wong, L.
Atoms
2,476
Residues
254
Protein chains
2
Unmodeled fraction
7.97%

Evaluations

R-work
0.185
R-free
0.237
Clashscore
6.1

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
PROTEIN (UROKINASE-TYPE PLASMINOGEN ACTIVATOR)23
  • ConstructSHORT CHAIN
Entity 2
MoleculeChainsLengthOrganismUniProtDetails
PROTEIN (UROKINASE-TYPE PLASMINOGEN ACTIVATOR)253
  • ConstructCATALYTIC DOMAIN

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations