Ensemble refinement model

PDB 3RWQ|dpdb_cen2ez22

Ensemble refinement model

Discovery of a Novel, Potent and Selective Inhibitor of 3-Phosphoinositide Dependent Kinase (PDK1)

Program
PHENIX phenix.ensemble_refinement
Model type
Ensemble
Purpose
Refinement
Atoms
99,279
Residues
283
Protein chains
1
Alternate-location fraction
0%
Ligands
3RW, GOL, SEP, SO4

Evaluations

R-work
0.159
R-free
0.228
Clashscore
—

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
3-phosphoinositide-dependent protein kinase 1311
  • ConstructKinase domain, residues 51-359

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations