Ensemble refinement model

PDB 3OW4|dpdb_ck6nmmzz

Ensemble refinement model

Discovery of dihydrothieno- and dihydrofuropyrimidines as potent pan Akt inhibitors

Program
PHENIX phenix.ensemble_refinement
Model type
Ensemble
Purpose
Refinement
Atoms
188,435
Residues
654
Protein chains
4
Alternate-location fraction
0%
Ligands
SMY, TPO

Evaluations

R-work
0.166
R-free
0.225
Clashscore
—

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
RAC-alpha serine/threonine-protein kinase341
  • MutationS473D
Entity 2
MoleculeChainsLengthOrganismUniProtDetails
GSK 3 beta peptide10—

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations