Deposited model

PDB 7UZN|dpdb_foi5m76t

Deposited model

CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH BMT-206059 AKA 2-{(3M)-3-(1,4-DIMETHYL-1H-1,2,3-TRIAZOL-5-YL)-8-FLUORO-5-[(S)-(OXAN-4-YL)(PHENYL)METHYL]-5H-PYRIDO[3,2-b]INDOL-7-YL}PROPAN-2-OL, TRIPLY DEUTERATED ON THE 4-METHYL GROUP

Program
BUSTER 2.11.8 (3-FEB-2022)
Model type
Deposited
Purpose
Reference
Authors
Sheriff, S.
Atoms
1,161
Residues
125
Protein chains
1
Unmodeled fraction
2.34%
Ligand
NA

Evaluations

R-work
0.197
R-free
0.217
Clashscore
0.9

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Bromodomain-containing protein 4128
  • Constructfirst bromodomain

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations