Deposited model

PDB 1GJC|dpdb_fy1ldzue

Deposited model

ENGINEERING INHIBITORS HIGHLY SELECTIVE FOR THE S1 SITES OF SER190 TRYPSIN-LIKE SERINE PROTEASE DRUG TARGETS

Program
X-PLOR 3.851
Model type
Deposited
Purpose
Reference
Authors
Katz, B.A., Sprengeler, P.A., Luong, C., Verner, E., Spencer, J.R., Breitenbucher, J.G., Hui, H., McGee, D., Allen, D., Martelli, A., Mackman, R.L.
Atoms
2,358
Residues
255
Protein chains
2
Unmodeled fraction
7.61%
Ligand
CIT

Evaluations

R-work
0.199
R-free
0.242
Clashscore
7.3

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
UROKINASE-TYPE PLASMINOGEN ACTIVATOR23
  • ConstructSHORT CHAIN
Entity 2
MoleculeChainsLengthOrganismUniProtDetails
UROKINASE-TYPE PLASMINOGEN ACTIVATOR253
  • ConstructCATALYTIC DOMAIN
  • MutationN145A

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations