Deposited model

PDB 4C66|dpdb_g5pb77sv

Deposited model

Discovery of Epigenetic Regulator I-BET762: Lead Optimization to Afford a Clinical Candidate Inhibitor of the BET Bromodomains

Program
REFMAC 5.6.0117
Model type
Deposited
Purpose
Reference
Authors
Chung, C., Mirguet, O.
Atoms
1,190
Residues
126
Protein chains
1
Unmodeled fraction
0%

Evaluations

R-work
0.217
R-free
0.266
Clashscore
8.9

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
BROMODOMAIN-CONTAINING PROTEIN 4126
  • ConstructN-TERMINAL BROMODOMAIN, RESIDUES 44-167

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations