Deposited model

PDB 3QRK|dpdb_gg9teulb

Deposited model

The crystal structure of human abl1 kinase domain in complex with DP-987

Program
REFMAC 5.2.0005
Model type
Deposited
Purpose
Reference
Authors
Chan, W.W., Wise, S.C., Kaufman, M.D., Ahn, Y.M., Ensinger, C.L., Haack, T., Hood, M.M., Jones, J., Lord, J.W., Lu, W.P., Miller, D., Patt, W.C., Smith, B.D., Petillo, P.A., Rutkoski, T.J., Telikepalli, H., Vogeti, L., Yao, T., Chun, L., Clark, R., Evangelista, P., Gavrilescu, L.C., Lazarides, K., Zaleskas, V.M., Stewart, L.J., Van Etten, R.A., Flynn, D.L.
Atoms
2,357
Residues
270
Protein chains
1
Unmodeled fraction
2.53%

Evaluations

R-work
0.188
R-free
0.281
Clashscore
8.2

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Tyrosine-protein kinase ABL1277
  • ConstructKinase domain, UNP residues 229-499

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations