Deposited model

PDB 5DLX|dpdb_gsqwjjzw

Deposited model

FIRST DOMAIN OF HUMAN BROMODOMAIN BRD4 IN COMPLEX WITH INHIBITOR N-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}-1-{3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}piperidine-4-carboxamide

Program
REFMAC 5.8.0131
Model type
Deposited
Purpose
Reference
Authors
Raux, B., Rebuffet, E., Betzi, S., Morelli, X.
Atoms
1,115
Residues
125
Protein chains
1
Unmodeled fraction
1.57%

Evaluations

R-work
0.125
R-free
0.207
Clashscore
0.9

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Bromodomain-containing protein 4127
  • ConstructN-TERMINAL BROMODOMAIN, RESIDUES 42-168

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations