Deposited model

PDB 3E63|dpdb_i22kvwbm

Deposited model

Fragment based discovery of JAK-2 inhibitors

Program
REFMAC
Model type
Deposited
Purpose
Reference
Authors
Antonysamy, S., Fang, W., Hirst, G., Park, F., Russell, M., Smyth, L., Sprengeler, P., Stappenbeck, F., Steensma, R., Thompson, D.A., Wilson, M., Wong, M., Zhang, A., Zhang, F.
Atoms
2,695
Residues
292
Protein chains
1
Unmodeled fraction
0.34%

Evaluations

R-work
0.199
R-free
0.263
Clashscore
1.4

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Tyrosine-protein kinase JAK2293
  • ConstructCATALYTIC DOMAIN (UNP residues 839 to 1131)

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations