Deposited model

PDB 1GI8|dpdb_mfhg3g8k

Deposited model

A NOVEL SERINE PROTEASE INHIBITION MOTIF INVOLVING A MULTI-CENTERED SHORT HYDROGEN BONDING NETWORK AT THE ACTIVE SITE

Program
X-PLOR 3.851
Model type
Deposited
Purpose
Reference
Authors
Katz, B.A., Elrod, K., Luong, C., Rice, M., Mackman, R.L., Sprengeler, P.A., Spencer, J., Hatayte, J., Janc, J., Link, J., Litvak, J., Rai, R., Rice, K., Sideris, S., Verner, E., Young, W.
Atoms
2,473
Residues
254
Protein chains
2
Unmodeled fraction
5.22%
Ligand
CIT

Evaluations

R-work
0.200
R-free
0.254
Clashscore
9.6

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
UROKINASE-TYPE PLASMINOGEN ACTIVATOR23
  • ConstructSHORT CHAIN
Entity 2
MoleculeChainsLengthOrganismUniProtDetails
UROKINASE-TYPE PLASMINOGEN ACTIVATOR245
  • ConstructCATALYTIC DOMAIN
  • MutationN145A

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations