Deposited model

PDB 4CFM|dpdb_olqhz0yn

Deposited model

Structure-based design of C8-substituted O6-cyclohexylmethoxyguanine CDK1 and 2 inhibitors.

Program
REFMAC 5.8.0049
Model type
Deposited
Purpose
Reference
Authors
Carbain, B., Paterson, D.J., Anscombe, E., Campbell, A., Cano, C., Echalier, A., Endicott, J., Golding, B.T., Haggerty, K., Hardcastle, I.R., Jewsbury, P., Newell, D.R., Noble, M.E.M., Roche, C., Wang, L.Z., Griffin, R.
Atoms
8,829
Residues
1,080
Protein chains
4
Unmodeled fraction
3.74%

Evaluations

R-work
0.217
R-free
0.258
Clashscore
12.3

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
CYCLIN-DEPENDENT KINASE 2303—
Entity 2
MoleculeChainsLengthOrganismUniProtDetails
CYCLIN-A2258
  • ConstructCDK-ACTIVATING FRAGMENT, RESIDUES 175-432

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations