Deposited model

PDB 3E64|dpdb_ong70tkb

Deposited model

Fragment based discovery of JAK-2 inhibitors

Program
REFMAC
Model type
Deposited
Purpose
Reference
Authors
Antonysamy, S., Fang, W., Hirst, G., Park, F., Russell, M., Smyth, L., Sprengeler, P., Stappenbeck, F., Steensma, R., Thompson, D.A., Wilson, M., Wong, M., Zhang, A., Zhang, F.
Atoms
2,778
Residues
293
Protein chains
1
Unmodeled fraction
0%

Evaluations

R-work
0.169
R-free
0.220
Clashscore
2.9

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Tyrosine-protein kinase JAK2293
  • ConstructCATALYTIC DOMAIN (UNP residues 839 to 1131)

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations