Deposited model

PDB 6GDM|dpdb_p3grfrb6

Deposited model

Fragment-based discovery of a highly potent, orally bioavailable inhibitor which modulates the phosphorylation and catalytic activity of ERK1/2

Program
REFMAC 5.8.0222
Model type
Deposited
Purpose
Reference
Authors
O'Reilly, M.
Atoms
3,295
Residues
345
Protein chains
1
Unmodeled fraction
6.25%

Evaluations

R-work
0.182
R-free
0.243
Clashscore
4.5

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Mitogen-activated protein kinase 1368—

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations