Ensemble refinement model

PDB 4AG8|dpdb_q8ma55c9

Ensemble refinement model

CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH AXITINIB (AG-013736) (N-Methyl-2-(3-((E)-2-pyridin-2-yl-vinyl)-1H- indazol-6-ylsulfanyl)-benzamide)

Program
PHENIX phenix.ensemble_refinement
Model type
Ensemble
Purpose
Refinement
Atoms
103,736
Residues
296
Protein chains
1
Alternate-location fraction
0%
Ligand
AXI

Evaluations

R-work
0.160
R-free
0.200
Clashscore
—

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2316
  • ConstructKINASE DOMAIN, RESIDUES 806-940,990-1171
  • MutationsYES

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations