Deposited model

PDB 1C5O|dpdb_qyty3usm

Deposited model

STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR

Program
X-PLOR 3.1
Model type
Deposited
Purpose
Reference
Authors
Katz, B.A., Mackman, R., Luong, C., Radika, K., Martelli, A., Sprengeler, P.A., Wang, J., Chan, H., Wong, L.
Atoms
2,873
Residues
299
Protein chains
3
Unmodeled fraction
2.29%
Ligand
NA

Evaluations

R-work
0.200
R-free
0.262
Clashscore
5.5

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Thrombin light chain36
  • ConstructLIGHT CHAIN
Entity 2
MoleculeChainsLengthOrganismUniProtDetails
Thrombin heavy chain259
  • ConstructHEAVY CHAIN
Entity 3
MoleculeChainsLengthOrganismUniProtDetails
Hirudin11
  • Hirudo medicinalis6421
—

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations