Deposited model

PDB 4D0X|dpdb_suer1pji

Deposited model

Pyrrole-3-carboxamides as potent and selective JAK2 inhibitors

Program
REFMAC 5.6.0117
Model type
Deposited
Purpose
Reference
Authors
Canevari, G., Fasolini, M., Bertrand, J., Brasca, M.G., Nesi, M., Avanzi, N., Ballinari, D., Bandiera, T., Bindi, S., Carenzi, D., Casero, D., Ceriani, L., Ciomei, M., Cirla, A., Colombo, M., Cribioli, S., Cristiani, C., Della Vedova, F., Fachin, G., Felder, E.R., Galvani, A., Isacchi, A., Mirizzi, D., Motto, I., Panzeri, A., Pesenti, E., Vianello, P., Gnocchi, P., Donati, D.
Atoms
2,700
Residues
293
Protein chains
1
Unmodeled fraction
1.68%

Evaluations

R-work
0.163
R-free
0.219
Clashscore
6.7

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
TYROSINE-PROTEIN KINASE JAK2298
  • ConstructKINASE DOMAIN, RESIDUES 835-1132

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations