Deposited model

PDB 3QCY|dpdb_u4br8z21

Deposited model

Phosphoinositide-Dependent Kinase-1 (PDK1) kinase domain with 4-[2-Amino-6-(3-amino-1H-indazol-6-yl)-4-pyrimidinyl]-N-phenyl-2-morpholinecarboxamide

Program
REFMAC
Model type
Deposited
Purpose
Reference
Authors
Medina, J.R., Becker, C.J., Blackledge, C.W., Duquenne, C., Feng, Y., Grant, S.W., Heerding, D., Li, W.H., Miller, W.H., Romeril, S.P., Scherzer, D., Shu, A., Bobko, M.A., Chadderton, A.R., Dumble, M., Gradiner, C.M., Gilbert, S., Liu, Q., Rabindran, S.K., Sudakin, V., Xiang, H., Brady, P.G., Campobasso, N., Ward, P., Axten, J.M.
Atoms
2,398
Residues
275
Protein chains
1
Unmodeled fraction
11.86%

Evaluations

R-work
0.178
R-free
0.212
Clashscore
5.4

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
3-phosphoinositide-dependent protein kinase 1312
  • Constructkinase domain, residues 48-359

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations