Deposited model

PDB 5ACC|dpdb_ur52tsvj

Deposited model

A Novel Oral Selective Estrogen Receptor Down-regulator, AZD9496, drives Tumour Growth Inhibition in Estrogen Receptor positive and ESR1 Mutant Models

Program
REFMAC 5.8.0103
Model type
Deposited
Purpose
Reference
Authors
Norman, R.A., Weir, H.M., Bradbury, R.H., Lawson, M., Rabow, A.A., Buttar, D., Callis, R.J., Curwen, J.O., de Almeida, C., Ballard, P., Hulse, M., Donald, C.S., Feron, L.J.L., Gingell, H., Karoutchi, G., MacFaul, P., Moss, T., Pearson, S.E., Tonge, M., Davies, G., Walker, G.E., Wilson, Z., Rowlinson, R., Powell, S., Hemsley, P., Linney, E., Campbell, H., Ghazoui, Z., Sadler, C., Richmond, G., Pazolli, E., Mazzola, A.M., DCruz, C., De Savi, C.
Atoms
1,911
Residues
228
Protein chains
1
Unmodeled fraction
8.06%

Evaluations

R-work
0.217
R-free
0.266
Clashscore
1.9

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
ESTROGEN RECEPTOR248
  • ConstructLIGAND-BINDING DOMAIN, UNP RESIDUES 307-554
  • MutationsYES

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations