Deposited model

PDB 1UYL|dpdb_v3iec8a8

Deposited model

Structure-Activity Relationships in purine-based inhibitor binding to HSP90 isoforms

Program
REFMAC 5.0
Model type
Deposited
Purpose
Reference
Authors
Wright, L., Barril, X., Dymock, B., Sheridan, L., Surgenor, A., Beswick, M., Drysdale, M., Collier, A., Massey, A., Davies, N., Fink, A., Fromont, C., Aherne, W., Boxall, K., Sharp, S., Workman, P., Hubbard, R.E.
Atoms
1,922
Residues
208
Protein chains
1
Unmodeled fraction
11.86%

Evaluations

R-work
0.199
R-free
0.227
Clashscore
7.6

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
HEAT SHOCK PROTEIN HSP 90-ALPHA236
  • ConstructN-TERMINAL DOMAIN, RESIDUES 1-235

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations