Deposited model

PDB 3ZTX|dpdb_weksn244

Deposited model

Aurora kinase selective inhibitors identified using a Taxol-induced checkpoint sensitivity screen.

Program
REFMAC 5.5.0072
Model type
Deposited
Purpose
Reference
Authors
Kwiatkowski, N., Villa, F., Musacchio, A., Gray, N.
Atoms
5,567
Residues
626
Protein chains
4
Unmodeled fraction
4.57%

Evaluations

R-work
0.186
R-free
0.226
Clashscore
8.2

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
SERINE/THREONINE-PROTEIN KINASE 12-A284
  • ConstructKINASE DOMAIN, RESIDUES 78-361
Entity 2
MoleculeChainsLengthOrganismUniProtDetails
INNER CENTROMERE PROTEIN A44
  • ConstructRESIDUES 797-840

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations