Deposited model

PDB 5HKM|dpdb_y2h2jqqc

Deposited model

DISCOVERY OF NOVEL 7-AZAINDOLES AS PDK1 INHIBITORS

Program
BUSTER 2.11.6
Model type
Deposited
Purpose
Reference
Authors
Wucherer-Plietker, M., Esdar, C., Knoechel, T., Hillertz, P., Heinrich, T., Buchstaller, H.P., Greiner, H., Dorsch, D., Calderini, M., Bruge, D., Mueller, T.J.J., Graedler, U.
Atoms
2,345
Residues
273
Protein chains
1
Unmodeled fraction
11.65%

Evaluations

R-work
0.190
R-free
0.273
Clashscore
4.9

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
3-phosphoinositide-dependent protein kinase 1309
  • ConstructKINASE DOMAIN, RESIDUES 51-359

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations