Deposited model

PDB 6HRP|dpdb_yg9dty6b

Deposited model

CRYSTAL STRUCTURE OF BTK KINASE DOMAIN COMPLEXED WITH 6-(dimethylamino)-2-[2-(hydroxymethyl)-3-[1-methyl-5-[[5-(morpholine-4-carbonyl)-2-pyridyl]amino]-6-oxo-3-pyridyl]phenyl]-3,4-dihydroisoquinolin-1-one

Program
REFMAC 5.5.0072
Model type
Deposited
Purpose
Reference
Authors
Janson, C., Kuglstatter, A.
Atoms
2,630
Residues
263
Protein chains
1
Unmodeled fraction
7.07%

Evaluations

R-work
0.174
R-free
0.192
Clashscore
4.9

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Tyrosine-protein kinase BTK283
  • MutationsM489A R492A E624A K625A

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations