Deposited model

PDB 4D0W|dpdb_yzc8h9a3

Deposited model

Pyrrole-3-carboxamides as potent and selective JAK2 inhibitors

Program
REFMAC 5.6.0117
Model type
Deposited
Purpose
Reference
Authors
Bertrand, J., Canevari, G., Fasolini, M., Brasca, M.G., Nesi, M., Avanzi, N., Ballinari, D., Bandiera, T., Bindi, S., Carenzi, D., Casero, D., Ceriani, L., Ciomei, M., Cirla, A., Colombo, M., Cribioli, S., Cristiani, C., Della Vedova, F., Fachin, G., Felder, E.R., Galvani, A., Isacchi, A., Mirizzi, D., Motto, I., Panzeri, A., Pesenti, E., Vianello, P., Gnocchi, P., Donati, D.
Atoms
2,627
Residues
291
Protein chains
1
Unmodeled fraction
2.35%

Evaluations

R-work
0.173
R-free
0.215
Clashscore
8.5

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
TYROSINE-PROTEIN KINASE JAK2298
  • ConstructKINASE DOMAIN, RESIDUES 835-1132

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations