Deposited model

PDB 1C5X|dpdb_zacgza8n

Deposited model

STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR

Program
X-PLOR 3.1
Model type
Deposited
Purpose
Reference
Authors
Katz, B.A., Mackman, R., Luong, C., Radika, K., Martelli, A., Sprengeler, P.A., Wang, J., Chan, H., Wong, L.
Atoms
2,534
Residues
257
Protein chains
2
Unmodeled fraction
6.88%

Evaluations

R-work
0.195
R-free
0.244
Clashscore
5.2

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
PROTEIN (UROKINASE-TYPE PLASMINOGEN ACTIVATOR)23
  • ConstructSHORT CHAIN
Entity 2
MoleculeChainsLengthOrganismUniProtDetails
PROTEIN (UROKINASE-TYPE PLASMINOGEN ACTIVATOR)253
  • ConstructCATALYTIC DOMAIN

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations