Rerefined model

PDB 1GJB|dpdb_1k2grpdt

Rerefined model

ENGINEERING INHIBITORS HIGHLY SELECTIVE FOR THE S1 SITES OF SER190 TRYPSIN-LIKE SERINE PROTEASE DRUG TARGETS

Program
PHENIX 2.0_5824
Model type
Multiconformer
Purpose
Refinement
Atoms
2,217
Residues
254
Protein chains
2
Alternate-location fraction
1.97%
Ligands
130, CIT

Evaluations

R-work
0.213
R-free
0.270
Clashscore
11.5

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
UROKINASE-TYPE PLASMINOGEN ACTIVATOR23
  • ConstructSHORT CHAIN
Entity 2
MoleculeChainsLengthOrganismUniProtDetails
UROKINASE-TYPE PLASMINOGEN ACTIVATOR253
  • ConstructCATALYTIC DOMAIN
  • MutationN145A

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations