qFit model

PDB 1GJB|dpdb_1k2grpdt

qFit model

ENGINEERING INHIBITORS HIGHLY SELECTIVE FOR THE S1 SITES OF SER190 TRYPSIN-LIKE SERINE PROTEASE DRUG TARGETS

Program
Phenix 2.0_5824
Model type
Multiconformer
Purpose
Model Building
Atoms
5,267
Residues
234
Protein chains
2
Alternate-location fraction
95.3%
Ligands
130, CIT

Evaluations

R-work
0.213
R-free
0.304
Clashscore
—

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
UROKINASE-TYPE PLASMINOGEN ACTIVATOR23
  • ConstructSHORT CHAIN
Entity 2
MoleculeChainsLengthOrganismUniProtDetails
UROKINASE-TYPE PLASMINOGEN ACTIVATOR253
  • ConstructCATALYTIC DOMAIN
  • MutationN145A

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations