Deposited model

PDB 6TPD|dpdb_1tagfxcg

Deposited model

Fragment-based discovery of pyrazolopyridones as JAK1 inhibitors with excellent subtype selectivity

Program
REFMAC 5.8.0258
Model type
Deposited
Purpose
Reference
Authors
Hansen, B.B., Jepsen, T.J., Larsen, M., Sindet, R., Vifian, T., Burhardt, M.N., Larsen, J., Seitzberg, J.G., Carnerup, M.A., Jerre, A., Moelck, C., Rai, S., Nasipireddy, V.R., Ritzen, A.
Atoms
2,523
Residues
289
Protein chains
1
Unmodeled fraction
0%

Evaluations

R-work
0.223
R-free
0.278
Clashscore
4.0

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Tyrosine-protein kinase JAK2289
  • MutationsY1007F/Y1008F

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations