qFit model

PDB 6FEX|dpdb_8wn1751q

qFit model

DDR1, 2-[4-bromo-2-oxo-1'-(1H-pyrazolo[4,3-b]pyridine-5-carbonyl)spiro[indole-3,4'-piperidine]-1-yl]-N-(2,2,2-trifluoroethyl)acetamide, 1.291A, P212121, Rfree=17.4%

Program
Phenix 2.0_5824
Model type
Multiconformer
Purpose
Model Building
Atoms
4,706
Residues
289
Protein chains
1
Alternate-location fraction
67.82%
Ligands
CL, D6Z, IOD, MES

Evaluations

R-work
0.159
R-free
0.182
Clashscore
—

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Epithelial discoidin domain-containing receptor 1321
  • Constructtyrosine kinase domain, residues 593-913
  • MutationsDEL(730-735) 2-[4-bromo-2-oxo-1'-(1H-pyrazolo[4,3-b]pyridine-5-carbonyl)spiro[indole-3,4'-piperidine]-1-yl]-N-(2,2,2-trifluoroethyl)acetamide

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations