Deposited model

PDB 3RWQ|dpdb_cen2ez22

Deposited model

Discovery of a Novel, Potent and Selective Inhibitor of 3-Phosphoinositide Dependent Kinase (PDK1)

Program
REFMAC
Model type
Deposited
Purpose
Reference
Authors
Kazmirski, S., Kohls, D.
Atoms
2,467
Residues
284
Protein chains
1
Unmodeled fraction
8.68%

Evaluations

R-work
0.193
R-free
0.256
Clashscore
7.1

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
3-phosphoinositide-dependent protein kinase 1311
  • ConstructKinase domain, residues 51-359

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations