Deposited model

PDB 4I5M|dpdb_dwkb3wz9

Deposited model

Selective & Brain-Permeable Polo-like Kinase-2 (Plk-2) Inhibitors that Reduce -Synuclein Phosphorylation in Rat Brain

Program
REFMAC 5.2.0019
Model type
Deposited
Purpose
Reference
Authors
Aubele, D.L., Hom, R.K., Adler, M., Galemmo Jr., R.A., Bowers, S., Truong, A.P., Pan, H., Beroza, P., Neitz, R.J., Yao, N., Lin, M., Tonn, G., Zhang, H., Bova, M.P., Ren, Z., Tam, D., Ruslim, L., Baker, J., Diep, L., Fitzgerald, K., Hoffman, J., Motter, R., Fauss, D., Tanaka, P., Dappen, M., Jagodzinski, J., Chan, W., Konradi, A.W., Latimer, L., Zhu, Y.L., Artis, D.R., Sham, H.L., Anderson, J.P., Bergeron, M.
Atoms
2,533
Residues
273
Protein chains
1
Unmodeled fraction
11.36%

Evaluations

R-work
0.320
R-free
0.392
Clashscore
23.4

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Serine/threonine-protein kinase PLK2308
  • ConstructPLK2 kinase domain
  • MutationsC83S V87T A119S A216S C259A C291S L335T

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations