Deposited model

PDB 5TO8|dpdb_gps8bk71

Deposited model

Selectivity switch between FAK and Pyk2: Macrocyclization of FAK inhibitors improves Pyk2 potency

Program
PHENIX 1.8.2_1309
Model type
Deposited
Purpose
Reference
Authors
Newby, Z.E.
Atoms
2,049
Residues
250
Protein chains
1
Unmodeled fraction
11.35%

Evaluations

R-work
0.203
R-free
0.235
Clashscore
3.1

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
Protein-tyrosine kinase 2-beta282
  • ConstructUNP Residues 414-692

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations