Deposited model

PDB 4AG8|dpdb_q8ma55c9

Deposited model

CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH AXITINIB (AG-013736) (N-Methyl-2-(3-((E)-2-pyridin-2-yl-vinyl)-1H- indazol-6-ylsulfanyl)-benzamide)

Program
REFMAC 5.1.24
Model type
Deposited
Purpose
Reference
Authors
McTigue, M., Wickersham, J., Pinko, C., Kania, R.S., Bender, S.
Atoms
2,735
Residues
296
Protein chains
1
Unmodeled fraction
6.33%

Evaluations

R-work
0.195
R-free
0.241
Clashscore
3.5

Macromolecules

The same in every model of this entry.

Entity 1
MoleculeChainsLengthOrganismUniProtDetails
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 2316
  • ConstructKINASE DOMAIN, RESIDUES 806-940,990-1171
  • MutationsYES

Data

L0 Raw
L1 Processed
L2 Models
L3 Evaluations